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Metabolic stability
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Keyword
keyword
Metabolic stability
RIS
0.001
(Research Intensity Score)
Papers
200
Top papers
Bioisosteres of the Phenyl Ring: Recent Strategic Applications in Lead Optimization and Drug Design
2021 · 689 citations
Fluorine in the Pharmaceutical Industry: FDA‐Approved Fluorine‐Containing Drugs in 2024
2025 · 91 citations
Catalytic Asymmetric Synthesis of Chiral Caged Hydrocarbons as Arenes Bioisosteres
2025 · 68 citations
Chemistry and Pharmacology of Fluorinated Drugs Approved by the FDA (2016–2022)
2023 · 141 citations
A Fruitful Decade of Organofluorine Chemistry: New Reagents and Reactions
2022 · 259 citations
Activating cGAS-STING pathway with ROS-responsive nanoparticles delivering a hybrid prodrug for enhanced chemo-immunotherapy
2022 · 166 citations
Assembly of (hetero)aryl sulfilimines via copper-catalyzed enantioselective S-arylation of sulfenamides with (hetero)aryl Iodides
2025 · 32 citations
Flavonoids, Chalcones, and Their Fluorinated Derivatives—Recent Advances in Synthesis and Potential Medical Applications
2025 · 20 citations
Thianthrenium-enabled modular synthesis of bicyclo[1.1.1]pentanes
2025 · 19 citations
Newest papers
Metabolic Stability of Fluorinated Small Molecules: A Physical Organic Chemistry Perspective
2026 · 10 citations
Fluorine-containing FDA-approved small-molecule drugs in 2025: significance, synthetic insights, and therapeutic applications
2026 · 8 citations
Halogen-Containing Drugs in 2025: A Record Year for the Therapeutic Use and Synthesis of FDA-Approved Small Molecules
2026 · 6 citations
Therapeutic potential of Sheng-Xian-Tang in doxorubicin-induced chronic heart failure by regulation of phenylalanine metabolism disruption
2026 · 3 citations
Modular Access to α ‐Tertiary Amines: Electrochemical Tandem Di‐Functionalization of Olefins With Ammonia Surrogates and Amino Acids
2026
Atropisomeric Properties of N-Aryl 5H-dibenz[b,f]azepines
2026
FAP-Inhibitor Homodimers with Engineered Linker-SpacerUnits: Toward Optimized Radiopharmaceuticals
2026
Synthesis, molecular docking and preliminary anticancer activity of product-C as a hybrid compound against PI3K
2026
FDA approved drug containing acetamide group- a mini review
2026
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